Research Output per year
Research Output 2016 2019
2019
Community assessment to advance computational prediction of cancer drug combinations in a pharmacogenomic screen
AstraZeneca-Sanger Drug Combination DREAM Consortium, 1 Dec 2019, In : Nature Communications. 10, 1, 2674.Research output: Contribution to Journal › Article › Academic › peer-review
Open Access
Pharmacogenetics
Drug Combinations
drugs
cancer
predictions
The Landscape of Atypical and Eukaryotic Protein Kinases
Kanev, G. K., de Graaf, C., de Esch, I. J. P., Leurs, R., Würdinger, T., Westerman, B. A. & Kooistra, A. J., Nov 2019, In : Trends in Pharmacological Sciences. 40, 11, p. 818-832 15 p.Research output: Contribution to Journal › Review article › Academic › peer-review
Open Access
Protein Kinases
Phosphotransferases
Spine
Single Nucleotide Polymorphism
Tumors
2017
1.15 - Structural Chemogenomics Databases to Navigate Protein–Ligand Interaction Space
Kanev, G. K., Kooistra, A. J., de Esch, I. J. P. & de Graaf, C., 2017, 1.15 - Structural Chemogenomics Databases to Navigate Protein–Ligand Interaction Space. Comprehensive Medicinal Chemistry III ed. Elsvier, Vol. 1. p. 444-471Research output: Chapter in Book / Report / Conference proceeding › Chapter › Academic › peer-review
Ligands
Proteins
Proteome
Bioactivity
Data mining
2016
KLIFS: a structural kinase-ligand interaction database.
Kooistra, A. J., Kanev, G. K., van Linden, O. P. J., Leurs, R., de Esch, I. J. P. & de Graaf, C., 2016, In : Nucleic Acids Research. 44, D1, p. D365-D371Research output: Contribution to Journal › Article › Academic › peer-review
Open Access
Phosphotransferases
Databases
Ligands
Dermatoglyphics
Protein Kinases
PDEStrIAn: A phosphodiesterase structure and ligan interaction annotated database as a tool for structure-based drug design.
Jansen, C. J. W., Kooistra, A. J., Kanev, G. K., Leurs, R., de Esch, I. J. P. & de Graaf, C., 2016, In : Journal of Medicinal Chemistry. 59, 15, p. 7029-7065Research output: Contribution to Journal › Article › Academic › peer-review
Drug Design
Phosphoric Diester Hydrolases
Databases
Ligands
Dermatoglyphics