Bispyrimidines as potent histamine H4 receptor ligands: delineation of structure activity relationships and detailed H4 receptor binding mode

H. Engelhardt, S. Schultes, C. de Graaf, S. Nijmeijer, H.F. Vischer, O.B. Zuiderveld, J. Dobler, K. Stachurski, M. Mayer, H. Arnhof, D. Scharn, E.J.J. Haaksma, I.J.P. de Esch, R. Leurs

Research output: Contribution to JournalArticleAcademicpeer-review

Abstract

The basic methylpiperazine moiety is considered a necessary substructure for high histamine H
Original languageEnglish
Pages (from-to)4264-4276
JournalJournal of Medicinal Chemistry
Volume2013
Issue number56
DOIs
Publication statusPublished - 2013

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