Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist

H.D. Lim; R. van Rijn; P. Ling; R.A. Bakker; R.L. Thurmond; R. Leurs

doi:10.1124/jpet.105.087965

Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist

H.D. Lim, R. van Rijn, P. Ling, R.A. Bakker, R.L. Thurmond, R. Leurs

Medicinal chemistry

Research output: Contribution to Journal › Article › Academic › peer-review

Abstract

The histamine H

Original language	English
Pages (from-to)	1310-21
Journal	The Journal of Pharmacology and Experimental Therapeutics
Volume	314
Issue number	3
DOIs	https://doi.org/10.1124/jpet.105.087965
Publication status	Published - 2005

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10.1124/jpet.105.087965

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Lim, H. D., van Rijn, R., Ling, P., Bakker, R. A., Thurmond, R. L., & Leurs, R. (2005). Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist. The Journal of Pharmacology and Experimental Therapeutics, 314(3), 1310-21. https://doi.org/10.1124/jpet.105.087965

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title = "Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist",

abstract = "The histamine H",

author = "H.D. Lim and {van Rijn}, R. and P. Ling and R.A. Bakker and R.L. Thurmond and R. Leurs",

year = "2005",

doi = "10.1124/jpet.105.087965",

language = "English",

volume = "314",

pages = "1310--21",

journal = "The Journal of Pharmacology and Experimental Therapeutics",

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}

Lim, HD, van Rijn, R, Ling, P, Bakker, RA, Thurmond, RL & Leurs, R 2005, 'Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist', The Journal of Pharmacology and Experimental Therapeutics, vol. 314, no. 3, pp. 1310-21. https://doi.org/10.1124/jpet.105.087965

Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist. / Lim, H.D.; van Rijn, R.; Ling, P. et al.
In: The Journal of Pharmacology and Experimental Therapeutics, Vol. 314, No. 3, 2005, p. 1310-21.

Research output: Contribution to Journal › Article › Academic › peer-review

TY - JOUR

T1 - Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist

AU - Lim, H.D.

AU - van Rijn, R.

AU - Ling, P.

AU - Bakker, R.A.

AU - Thurmond, R.L.

AU - Leurs, R.

PY - 2005

Y1 - 2005

N2 - The histamine H

AB - The histamine H

U2 - 10.1124/jpet.105.087965

DO - 10.1124/jpet.105.087965

M3 - Article

SN - 0022-3565

VL - 314

SP - 1310

EP - 1321

JO - The Journal of Pharmacology and Experimental Therapeutics

JF - The Journal of Pharmacology and Experimental Therapeutics

IS - 3

ER -

Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist

Abstract

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