Abstract
The SAR of H3 ligands has been difficult to evaluate because of species differences, multiple isoforms and constitutive activity, among other complicating factors. A review is given of the sometimes-conflicting affinity, activity and efficacy data of H3 agonists that has been described in literature to date.
| Original language | English |
|---|---|
| Pages (from-to) | 955-63 |
| Number of pages | 9 |
| Journal | Mini-Reviews in Medicinal Chemistry |
| Volume | 4 |
| Issue number | 9 |
| DOIs | |
| Publication status | Published - Nov 2004 |
UN SDGs
This output contributes to the following UN Sustainable Development Goals (SDGs)
-
SDG 3 Good Health and Well-being
Keywords
- Animals
- Histamine Agonists
- Humans
- Ligands
- Receptors, Histamine H3
- Stereoisomerism
- Structure-Activity Relationship
- Journal Article
- Review
Fingerprint
Dive into the research topics of 'Histamine H3 receptor agonists'. Together they form a unique fingerprint.Cite this
- APA
- Author
- BIBTEX
- Harvard
- Standard
- RIS
- Vancouver