Homology modeling of rat and human cytochrome P450 2D (CYP2D) isoforms and computational rationalization of experimental ligand-binding specificities

J. Venhorst, A.M. ter Laak, J.N.M. Commandeur, Y. Funae, T. Hiroi, N.P.E. Vermeulen

Research output: Contribution to JournalArticleAcademicpeer-review

Abstract

The ligand-binding characteristics of rat and human CYP2D isoforms, i.e., rat CYP2D1-4 and human CYP2D6, were investigated by measuring IC
Original languageEnglish
Pages (from-to)74-86
JournalJournal of Medicinal Chemistry
Volume46
Issue number1
DOIs
Publication statusPublished - 2003

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