Human glutathione S-transferases- and NAD(P)H:quinone oxidoreductase 1-catalyzed inactivation of reactive quinoneimines of amodiaquine and N-desethylamodiaquine: Possible implications for susceptibility to amodiaquine-induced liver toxicity

Yongjie Zhang, Shalenie P den Braver-Sewradj, J Chris Vos, Nico P E Vermeulen, Jan N M Commandeur

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Pharmacology, Toxicology and Pharmaceutical Science