Synthesis and QSAR of quinazoline sulfonamides as highly potent human histamine H4 receptor inverse agonists.

R.A. Smits; M. Adami; E.P. Istyastono; O.P. Zuiderveld; C.M. Van Dam; F.J.J. De Kanter; A. Jongejan; G. Coruzzi; R. Leurs; I.J. De Esch

doi:10.1021/jm901379s

Synthesis and QSAR of quinazoline sulfonamides as highly potent human histamine H4 receptor inverse agonists.

R.A. Smits, M. Adami, E.P. Istyastono, O.P. Zuiderveld, C.M. Van Dam, F.J.J. De Kanter, A. Jongejan, G. Coruzzi, R. Leurs, I.J. De Esch

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Research output: Contribution to Journal › Article › Academic › peer-review

Abstract

Hit optimization of the class of quinazoline containing histamine H

Original language	English
Pages (from-to)	2390-2400
Journal	Journal of Medicinal Chemistry
Volume	53
DOIs	https://doi.org/10.1021/jm901379s
Publication status	Published - 2010

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10.1021/jm901379s

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@article{083d10d612d4448a9a16961ae13559c2,

title = "Synthesis and QSAR of quinazoline sulfonamides as highly potent human histamine H4 receptor inverse agonists.",

abstract = "Hit optimization of the class of quinazoline containing histamine H",

author = "R.A. Smits and M. Adami and E.P. Istyastono and O.P. Zuiderveld and \{Van Dam\}, C.M. and \{De Kanter\}, F.J.J. and A. Jongejan and G. Coruzzi and R. Leurs and \{De Esch\}, I.J.",

year = "2010",

doi = "10.1021/jm901379s",

language = "English",

volume = "53",

pages = "2390--2400",

journal = "Journal of Medicinal Chemistry",

issn = "0022-2623",

publisher = "American Chemical Society",

}

TY - JOUR

T1 - Synthesis and QSAR of quinazoline sulfonamides as highly potent human histamine H4 receptor inverse agonists.

AU - Smits, R.A.

AU - Adami, M.

AU - Istyastono, E.P.

AU - Zuiderveld, O.P.

AU - Van Dam, C.M.

AU - De Kanter, F.J.J.

AU - Jongejan, A.

AU - Coruzzi, G.

AU - Leurs, R.

AU - De Esch, I.J.

PY - 2010

Y1 - 2010

N2 - Hit optimization of the class of quinazoline containing histamine H

AB - Hit optimization of the class of quinazoline containing histamine H

UR - https://www.scopus.com/pages/publications/77949816697

UR - https://www.scopus.com/inward/citedby.url?scp=77949816697&partnerID=8YFLogxK

U2 - 10.1021/jm901379s

DO - 10.1021/jm901379s

M3 - Article

SN - 0022-2623

VL - 53

SP - 2390

EP - 2400

JO - Journal of Medicinal Chemistry

JF - Journal of Medicinal Chemistry

ER -

Synthesis and QSAR of quinazoline sulfonamides as highly potent human histamine H4 receptor inverse agonists.

Abstract

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