Synthesis, biological evaluation and automated docking of constrained analogs of the opioid peptide H-Dmt-D-AlapPhe-Gly-NH2 using the 4- or 5-metyl substsituted 4-amino-1,2,3,4-tetrahydro-2-benzazepin-3-one scaffold.

R de Wachter, C. de Graaf, C Keresztes, B Vandormael, S Ballet, G. Toth, D. Rognan, D Tourwé

Research output: Contribution to JournalArticleAcademicpeer-review

Original languageEnglish
Pages (from-to)3384-3393
Number of pages10
JournalJournal of Medicinal Chemistry
Publication statusPublished - 2011

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