Synthesis, biological evaluation, and automated docking of constrained analogues of the opioid peptide H-Dmt-d-Ala-Phe-Gly-NH 2 using the 4- or 5-methyl substituted 4-amino-1,2,4,5-tetrahydro-2-benzazepin-3-one scaffold

Rien De Wachter, Chris De Graaf*, Atilla Keresztes, Bart Vandormael, Steven Ballet, Géza Tóth, Didier Rognan, Dirk Tourwé

*Corresponding author for this work

Research output: Contribution to Journal › Article › Academic › peer-review

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Chemistry

Pharmacology, Toxicology and Pharmaceutical Science