Synthesis of 4-aminoquinolines by aerobic oxidative palladium-catalyzed double C-H activation and isocyanide insertion

T. Vlaar; B.U.W. Maes; E. Ruijter; R.V.A. Orru

doi:10.1007/s10593-013-1324-z

Synthesis of 4-aminoquinolines by aerobic oxidative palladium-catalyzed double C-H activation and isocyanide insertion

T. Vlaar
, B.U.W. Maes
, E. Ruijter
, R.V.A. Orru

AIMMS

Research output: Contribution to Journal › Article › Academic › peer-review

Abstract

An unprecedented aerobic oxidative Pd-catalyzed imidoylative coupling of two C-H fragments furnishing medicinally valuable 4-aminoquinolines is reported. Optimization studies are described and several analogs were successfully prepared. © 2013 Springer Science+Business Media New York.

Original language	English
Pages (from-to)	902-908
Journal	Chemistry of Heterocyclic Compounds
Volume	2013
Issue number	49
DOIs	https://doi.org/10.1007/s10593-013-1324-z
Publication status	Published - 2013

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title = "Synthesis of 4-aminoquinolines by aerobic oxidative palladium-catalyzed double C-H activation and isocyanide insertion",

abstract = "An unprecedented aerobic oxidative Pd-catalyzed imidoylative coupling of two C-H fragments furnishing medicinally valuable 4-aminoquinolines is reported. Optimization studies are described and several analogs were successfully prepared. {\textcopyright} 2013 Springer Science+Business Media New York.",

author = "T. Vlaar and B.U.W. Maes and E. Ruijter and R.V.A. Orru",

year = "2013",

doi = "10.1007/s10593-013-1324-z",

language = "English",

volume = "2013",

pages = "902--908",

journal = "Chemistry of Heterocyclic Compounds",

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TY - JOUR

T1 - Synthesis of 4-aminoquinolines by aerobic oxidative palladium-catalyzed double C-H activation and isocyanide insertion

AU - Vlaar, T.

AU - Maes, B.U.W.

AU - Ruijter, E.

AU - Orru, R.V.A.

PY - 2013

Y1 - 2013

N2 - An unprecedented aerobic oxidative Pd-catalyzed imidoylative coupling of two C-H fragments furnishing medicinally valuable 4-aminoquinolines is reported. Optimization studies are described and several analogs were successfully prepared. © 2013 Springer Science+Business Media New York.

AB - An unprecedented aerobic oxidative Pd-catalyzed imidoylative coupling of two C-H fragments furnishing medicinally valuable 4-aminoquinolines is reported. Optimization studies are described and several analogs were successfully prepared. © 2013 Springer Science+Business Media New York.

U2 - 10.1007/s10593-013-1324-z

DO - 10.1007/s10593-013-1324-z

M3 - Article

SN - 0009-3122

VL - 2013

SP - 902

EP - 908

JO - Chemistry of Heterocyclic Compounds

JF - Chemistry of Heterocyclic Compounds

IS - 49

ER -

Synthesis of 4-aminoquinolines by aerobic oxidative palladium-catalyzed double C-H activation and isocyanide insertion

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